Values CatLog read from this paper
Active-site mapping of bovine and human blood coagulation serine proteases using synthetic peptide 4-nitroanilide and thio ester substrates
PMID 6370301doi:10.1021/bi00299a009Open in Browse
The paper itself is not on this site: read it at the publisher. This page lists only the values CatLog read from it.
CatLog read 131 records (307 values) from this paper: activated protein C, β-factor XIIa, factor Xa and 3 more from Bos taurus, Homo sapiens.
Read from the paper by an AI model and checked against the paper by a second, separate AI run; code converted the units. Values are in CatLog's units; each record opens in Browse with the line the paper prints and the checks.
EC 3.4.21.6, EC 3.4.21.22, EC 3.4.21.27, EC 3.4.21.38
| Enzyme | Organism | Substrate | kcat (s⁻¹) | Km (mM) | kcat/Km (mM⁻¹ s⁻¹) | Conditions | Open record |
|---|---|---|---|---|---|---|---|
| activated protein C | Bos taurus | N-benzyloxycarbonyl-glycyl-L-arginine S-isobutyl thioester (SCH2CH(CH3)2) | 30 | 0.03 | 1 × 10³ | pH 7.5, 25 °C | Open record: activated protein C, N-benzyloxycarbonyl-glycyl-L-arginine S-isobutyl thioester (SCH2CH(CH3)2) |
| activated protein C | Bos taurus | N-benzyloxycarbonyl-L-alanyl-glycyl-L-arginine 4-nitroanilide | — | — | 3.4 | pH 8, 25 °C | Open record: activated protein C, N-benzyloxycarbonyl-L-alanyl-glycyl-L-arginine 4-nitroanilide |
| activated protein C | Bos taurus | N-benzyloxycarbonyl-L-alanyl-L-arginine S-benzyl thioester (SCH2C6H5) | 112 | 0.12 | 930 | pH 7.5, 25 °C | Open record: activated protein C, N-benzyloxycarbonyl-L-alanyl-L-arginine S-benzyl thioester (SCH2C6H5) |
| activated protein C | Bos taurus | N-benzyloxycarbonyl-L-alanyl-L-arginine S-isobutyl thioester (SCH2CH(CH3)2) | 47 | 0.052 | 900 | pH 7.5, 25 °C | Open record: activated protein C, N-benzyloxycarbonyl-L-alanyl-L-arginine S-isobutyl thioester (SCH2CH(CH3)2) |
| activated protein C | Bos taurus | N-benzyloxycarbonyl-L-alanyl-L-phenylalanyl-L-arginine 4-nitroanilide | 11 | 0.86 | 13 | pH 8, 25 °C | Open record: activated protein C, N-benzyloxycarbonyl-L-alanyl-L-phenylalanyl-L-arginine 4-nitroanilide |
| activated protein C | Bos taurus | N-benzyloxycarbonyl-L-alpha-glutamyl-glycyl-L-arginine 4-nitroanilide | — | — | 2.4 | pH 8, 25 °C | Open record: activated protein C, N-benzyloxycarbonyl-L-alpha-glutamyl-glycyl-L-arginine 4-nitroanilide |
| activated protein C | Bos taurus | N-benzyloxycarbonyl-L-alpha-glutamyl-L-arginine S-isobutyl thioester (SCH2CH(CH3)2) | 14 | 0.053 | 260 | pH 7.5, 25 °C | Open record: activated protein C, N-benzyloxycarbonyl-L-alpha-glutamyl-L-arginine S-isobutyl thioester (SCH2CH(CH3)2) |
| activated protein C | Bos taurus | N-benzyloxycarbonyl-L-alpha-glutamyl-L-phenylalanyl-L-arginine 4-nitroanilide | — | — | 8 | pH 8, 25 °C | Open record: activated protein C, N-benzyloxycarbonyl-L-alpha-glutamyl-L-phenylalanyl-L-arginine 4-nitroanilide |
| activated protein C | Bos taurus | N-benzyloxycarbonyl-L-arginine S-benzyl thioester (SCH2C6H5) | 39 | 0.036 | 1.1 × 10³ | pH 7.5, 25 °C | Open record: activated protein C, N-benzyloxycarbonyl-L-arginine S-benzyl thioester (SCH2C6H5) |
| activated protein C | Bos taurus | N-benzyloxycarbonyl-L-asparaginyl-glycyl-L-arginine 4-nitroanilide | 5 | 0.94 | 5.2 | pH 8, 25 °C | Open record: activated protein C, N-benzyloxycarbonyl-L-asparaginyl-glycyl-L-arginine 4-nitroanilide |
| activated protein C | Bos taurus | N-benzyloxycarbonyl-L-asparaginyl-L-phenylalanyl-L-arginine 4-nitroanilide | — | — | 22 | pH 8, 25 °C | Open record: activated protein C, N-benzyloxycarbonyl-L-asparaginyl-L-phenylalanyl-L-arginine 4-nitroanilide |
| activated protein C | Bos taurus | N-benzyloxycarbonyl-L-lysyl-glycyl-L-arginine 4-nitroanilide | 3.2 | 0.72 | 4.5 | pH 8, 25 °C | Open record: activated protein C, N-benzyloxycarbonyl-L-lysyl-glycyl-L-arginine 4-nitroanilide |
| activated protein C | Bos taurus | N-benzyloxycarbonyl-L-lysyl-L-arginine S-isobutyl thioester (SCH2CH(CH3)2) | 140 | 0.15 | 930 | pH 7.5, 25 °C | Open record: activated protein C, N-benzyloxycarbonyl-L-lysyl-L-arginine S-isobutyl thioester (SCH2CH(CH3)2) |
| activated protein C | Bos taurus | N-benzyloxycarbonyl-L-lysyl-L-phenylalanyl-L-arginine 4-nitroanilide | 5.5 | 0.37 | 15 | pH 8, 25 °C | Open record: activated protein C, N-benzyloxycarbonyl-L-lysyl-L-phenylalanyl-L-arginine 4-nitroanilide |
| activated protein C | Bos taurus | N-benzyloxycarbonyl-L-methionyl-L-arginine S-isobutyl thioester (SCH2CH(CH3)2) | 23 | 0.027 | 850 | pH 7.5, 25 °C | Open record: activated protein C, N-benzyloxycarbonyl-L-methionyl-L-arginine S-isobutyl thioester (SCH2CH(CH3)2) |
| activated protein C | Bos taurus | N-benzyloxycarbonyl-L-phenylalanyl-glycyl-L-arginine 4-nitroanilide | 3.8 | 3.3 | 1.1 | pH 8, 25 °C | Open record: activated protein C, N-benzyloxycarbonyl-L-phenylalanyl-glycyl-L-arginine 4-nitroanilide |
| activated protein C | Bos taurus | N-benzyloxycarbonyl-L-phenylalanyl-L-arginine S-isobutyl thioester (SCH2CH(CH3)2) | 81 | 0.011 | 740 | pH 7.5, 25 °C | Open record: activated protein C, N-benzyloxycarbonyl-L-phenylalanyl-L-arginine S-isobutyl thioester (SCH2CH(CH3)2) |
| activated protein C | Bos taurus | N-benzyloxycarbonyl-L-phenylalanyl-L-phenylalanyl-L-arginine 4-nitroanilide | — | — | 8.9 | pH 8, 25 °C | Open record: activated protein C, N-benzyloxycarbonyl-L-phenylalanyl-L-phenylalanyl-L-arginine 4-nitroanilide |
| activated protein C | Bos taurus | N-benzyloxycarbonyl-L-prolyl-glycyl-L-arginine 4-nitroanilide | — | — | 1.2 | pH 8, 25 °C | Open record: activated protein C, N-benzyloxycarbonyl-L-prolyl-glycyl-L-arginine 4-nitroanilide |
| activated protein C | Bos taurus | N-benzyloxycarbonyl-L-prolyl-L-arginine S-isobutyl thioester (SCH2CH(CH3)2) | 41 | 0.07 | 580 | pH 7.5, 25 °C | Open record: activated protein C, N-benzyloxycarbonyl-L-prolyl-L-arginine S-isobutyl thioester (SCH2CH(CH3)2) |
| activated protein C | Bos taurus | N-benzyloxycarbonyl-L-prolyl-L-phenylalanyl-L-arginine 4-nitroanilide | — | — | 1.8 | pH 8, 25 °C | Open record: activated protein C, N-benzyloxycarbonyl-L-prolyl-L-phenylalanyl-L-arginine 4-nitroanilide |
| activated protein C | Bos taurus | N-benzyloxycarbonyl-L-seryl-glycyl-L-arginine 4-nitroanilide | — | — | 5.4 | pH 8, 25 °C | Open record: activated protein C, N-benzyloxycarbonyl-L-seryl-glycyl-L-arginine 4-nitroanilide |
| activated protein C | Bos taurus | N-benzyloxycarbonyl-L-seryl-L-arginine S-isobutyl thioester (SCH2CH(CH3)2) | 30 | 0.083 | 360 | pH 7.5, 25 °C | Open record: activated protein C, N-benzyloxycarbonyl-L-seryl-L-arginine S-isobutyl thioester (SCH2CH(CH3)2) |
| activated protein C | Bos taurus | N-benzyloxycarbonyl-L-seryl-L-phenylalanyl-L-arginine 4-nitroanilide | — | — | 65 | pH 8, 25 °C | Open record: activated protein C, N-benzyloxycarbonyl-L-seryl-L-phenylalanyl-L-arginine 4-nitroanilide |
| activated protein C | Bos taurus | N-benzyloxycarbonyl-L-threonyl-L-arginine S-isobutyl thioester (SCH2CH(CH3)2) | 47 | 0.072 | 650 | pH 7.5, 25 °C | Open record: activated protein C, N-benzyloxycarbonyl-L-threonyl-L-arginine S-isobutyl thioester (SCH2CH(CH3)2) |
| activated protein C | Bos taurus | N-benzyloxycarbonyl-L-valyl-L-arginine S-isobutyl thioester (SCH2CH(CH3)2) | 25 | 0.044 | 570 | pH 7.5, 25 °C | Open record: activated protein C, N-benzyloxycarbonyl-L-valyl-L-arginine S-isobutyl thioester (SCH2CH(CH3)2) |
| activated protein C | Bos taurus | N-tert-butyloxycarbonyl-L-arginine S-benzyl thioester (SCH2C6H5) | 94 | 0.12 | 780 | pH 7.5, 25 °C | Open record: activated protein C, N-tert-butyloxycarbonyl-L-arginine S-benzyl thioester (SCH2C6H5) |
| activated protein C | Bos taurus | N-tert-butyloxycarbonyl-L-arginine S-isobutyl thioester (SCH2CH(CH3)2) | 41 | 0.048 | 850 | pH 7.5, 25 °C | Open record: activated protein C, N-tert-butyloxycarbonyl-L-arginine S-isobutyl thioester (SCH2CH(CH3)2) |
| activated protein C | Homo sapiens | N-benzyloxycarbonyl-glycyl-L-arginine S-isobutyl thioester (SCH2CH(CH3)2) | — | — | 48 | pH 8, 25 °C | Open record: activated protein C, N-benzyloxycarbonyl-glycyl-L-arginine S-isobutyl thioester (SCH2CH(CH3)2) |
| activated protein C | Homo sapiens | N-benzyloxycarbonyl-L-alanyl-glycyl-L-arginine 4-nitroanilide | — | — | 0.029 | pH 8, 25 °C | Open record: activated protein C, N-benzyloxycarbonyl-L-alanyl-glycyl-L-arginine 4-nitroanilide |
| activated protein C | Homo sapiens | N-benzyloxycarbonyl-L-alanyl-L-arginine S-benzyl thioester (SCH2C6H5) | 18 | 0.18 | 98 | pH 8, 25 °C | Open record: activated protein C, N-benzyloxycarbonyl-L-alanyl-L-arginine S-benzyl thioester (SCH2C6H5) |
| activated protein C | Homo sapiens | N-benzyloxycarbonyl-L-alanyl-L-arginine S-isobutyl thioester (SCH2CH(CH3)2) | — | — | 36 | pH 8, 25 °C | Open record: activated protein C, N-benzyloxycarbonyl-L-alanyl-L-arginine S-isobutyl thioester (SCH2CH(CH3)2) |
| activated protein C | Homo sapiens | N-benzyloxycarbonyl-L-alanyl-L-phenylalanyl-L-arginine 4-nitroanilide | — | — | 1.3 | pH 8, 25 °C | Open record: activated protein C, N-benzyloxycarbonyl-L-alanyl-L-phenylalanyl-L-arginine 4-nitroanilide |
| activated protein C | Homo sapiens | N-benzyloxycarbonyl-L-alpha-glutamyl-glycyl-L-arginine 4-nitroanilide | — | — | 0.042 | pH 8, 25 °C | Open record: activated protein C, N-benzyloxycarbonyl-L-alpha-glutamyl-glycyl-L-arginine 4-nitroanilide |
| activated protein C | Homo sapiens | N-benzyloxycarbonyl-L-alpha-glutamyl-L-phenylalanyl-L-arginine 4-nitroanilide | 1.2 | 0.59 | 1.6 | pH 8, 25 °C | Open record: activated protein C, N-benzyloxycarbonyl-L-alpha-glutamyl-L-phenylalanyl-L-arginine 4-nitroanilide |
| activated protein C | Homo sapiens | N-benzyloxycarbonyl-L-arginine S-isobutyl thioester (SCH2CH(CH3)2) | — | — | 54 | pH 8, 25 °C | Open record: activated protein C, N-benzyloxycarbonyl-L-arginine S-isobutyl thioester (SCH2CH(CH3)2) |
| activated protein C | Homo sapiens | N-benzyloxycarbonyl-L-asparaginyl-glycyl-L-arginine 4-nitroanilide | 0.18 | 0.9 | 0.148 | pH 8, 25 °C | Open record: activated protein C, N-benzyloxycarbonyl-L-asparaginyl-glycyl-L-arginine 4-nitroanilide |
| activated protein C | Homo sapiens | N-benzyloxycarbonyl-L-asparaginyl-L-phenylalanyl-L-arginine 4-nitroanilide | — | — | 2.4 | pH 8, 25 °C | Open record: activated protein C, N-benzyloxycarbonyl-L-asparaginyl-L-phenylalanyl-L-arginine 4-nitroanilide |
| activated protein C | Homo sapiens | N-benzyloxycarbonyl-L-lysyl-glycyl-L-arginine 4-nitroanilide | 1.3 | 9.9 | 0.1 | pH 8, 25 °C | Open record: activated protein C, N-benzyloxycarbonyl-L-lysyl-glycyl-L-arginine 4-nitroanilide |
| activated protein C | Homo sapiens | N-benzyloxycarbonyl-L-lysyl-L-arginine S-isobutyl thioester (SCH2CH(CH3)2) | — | — | 50 | pH 8, 25 °C | Open record: activated protein C, N-benzyloxycarbonyl-L-lysyl-L-arginine S-isobutyl thioester (SCH2CH(CH3)2) |
| activated protein C | Homo sapiens | N-benzyloxycarbonyl-L-lysyl-L-phenylalanyl-L-arginine 4-nitroanilide | 7.9 | 1.8 | 3.2 | pH 8, 25 °C | Open record: activated protein C, N-benzyloxycarbonyl-L-lysyl-L-phenylalanyl-L-arginine 4-nitroanilide |
| activated protein C | Homo sapiens | N-benzyloxycarbonyl-L-methionyl-L-arginine S-isobutyl thioester (SCH2CH(CH3)2) | 4 | 0.79 | 5.6 | pH 8, 25 °C | Open record: activated protein C, N-benzyloxycarbonyl-L-methionyl-L-arginine S-isobutyl thioester (SCH2CH(CH3)2) |
| activated protein C | Homo sapiens | N-benzyloxycarbonyl-L-phenylalanyl-L-arginine S-isobutyl thioester (SCH2CH(CH3)2) | 4 | 0.032 | 120 | pH 8, 25 °C | Open record: activated protein C, N-benzyloxycarbonyl-L-phenylalanyl-L-arginine S-isobutyl thioester (SCH2CH(CH3)2) |
| activated protein C | Homo sapiens | N-benzyloxycarbonyl-L-phenylalanyl-L-phenylalanyl-L-arginine 4-nitroanilide | — | — | 0.6 | pH 8, 25 °C | Open record: activated protein C, N-benzyloxycarbonyl-L-phenylalanyl-L-phenylalanyl-L-arginine 4-nitroanilide |
| activated protein C | Homo sapiens | N-benzyloxycarbonyl-L-prolyl-L-arginine S-isobutyl thioester (SCH2CH(CH3)2) | 3 | 0.1 | 28 | pH 8, 25 °C | Open record: activated protein C, N-benzyloxycarbonyl-L-prolyl-L-arginine S-isobutyl thioester (SCH2CH(CH3)2) |
| activated protein C | Homo sapiens | N-benzyloxycarbonyl-L-prolyl-L-phenylalanyl-L-arginine 4-nitroanilide | — | — | 0.074 | pH 8, 25 °C | Open record: activated protein C, N-benzyloxycarbonyl-L-prolyl-L-phenylalanyl-L-arginine 4-nitroanilide |
| activated protein C | Homo sapiens | N-benzyloxycarbonyl-L-seryl-glycyl-L-arginine 4-nitroanilide | 0.16 | 1.6 | 0.073 | pH 8, 25 °C | Open record: activated protein C, N-benzyloxycarbonyl-L-seryl-glycyl-L-arginine 4-nitroanilide |
| activated protein C | Homo sapiens | N-benzyloxycarbonyl-L-seryl-L-arginine S-isobutyl thioester (SCH2CH(CH3)2) | — | — | 13 | pH 8, 25 °C | Open record: activated protein C, N-benzyloxycarbonyl-L-seryl-L-arginine S-isobutyl thioester (SCH2CH(CH3)2) |
| activated protein C | Homo sapiens | N-benzyloxycarbonyl-L-seryl-L-phenylalanyl-L-arginine 4-nitroanilide | — | — | 3.9 | pH 8, 25 °C | Open record: activated protein C, N-benzyloxycarbonyl-L-seryl-L-phenylalanyl-L-arginine 4-nitroanilide |
| activated protein C | Homo sapiens | N-benzyloxycarbonyl-L-threonyl-L-arginine S-isobutyl thioester (SCH2CH(CH3)2) | 4 | 0.1 | 44 | pH 8, 25 °C | Open record: activated protein C, N-benzyloxycarbonyl-L-threonyl-L-arginine S-isobutyl thioester (SCH2CH(CH3)2) |
| activated protein C | Homo sapiens | N-benzyloxycarbonyl-L-valyl-L-arginine S-isobutyl thioester (SCH2CH(CH3)2) | — | — | 53 | pH 8, 25 °C | Open record: activated protein C, N-benzyloxycarbonyl-L-valyl-L-arginine S-isobutyl thioester (SCH2CH(CH3)2) |
| activated protein C | Homo sapiens | N-tert-butyloxycarbonyl-L-arginine S-benzyl thioester (SCH2C6H5) | — | — | 74 | pH 8, 25 °C | Open record: activated protein C, N-tert-butyloxycarbonyl-L-arginine S-benzyl thioester (SCH2C6H5) |
| factor IXa | Bos taurus | N-benzyloxycarbonyl-L-alanyl-glycyl-L-arginine 4-nitroanilide | — | — | 0.015 | pH 7.5, 25 °C | Open record: factor IXa, N-benzyloxycarbonyl-L-alanyl-glycyl-L-arginine 4-nitroanilide |
| factor IXa | Bos taurus | N-benzyloxycarbonyl-L-alpha-glutamyl-glycyl-L-arginine 4-nitroanilide | — | — | 0.503 | pH 7.5, 25 °C | Open record: factor IXa, N-benzyloxycarbonyl-L-alpha-glutamyl-glycyl-L-arginine 4-nitroanilide |
| factor IXa | Bos taurus | N-benzyloxycarbonyl-L-alpha-glutamyl-L-phenylalanyl-L-arginine 4-nitroanilide | — | — | 0.0019 | pH 7.5, 25 °C | Open record: factor IXa, N-benzyloxycarbonyl-L-alpha-glutamyl-L-phenylalanyl-L-arginine 4-nitroanilide |
| factor IXa | Bos taurus | N-benzyloxycarbonyl-L-asparaginyl-glycyl-L-arginine 4-nitroanilide | — | — | 0.011 | pH 7.5, 25 °C | Open record: factor IXa, N-benzyloxycarbonyl-L-asparaginyl-glycyl-L-arginine 4-nitroanilide |
| factor IXa | Bos taurus | N-benzyloxycarbonyl-L-asparaginyl-L-phenylalanyl-L-arginine 4-nitroanilide | — | — | 0.0079 | pH 7.5, 25 °C | Open record: factor IXa, N-benzyloxycarbonyl-L-asparaginyl-L-phenylalanyl-L-arginine 4-nitroanilide |
| factor IXa | Bos taurus | N-benzyloxycarbonyl-L-lysyl-glycyl-L-arginine 4-nitroanilide | — | — | 0.0064 | pH 7.5, 25 °C | Open record: factor IXa, N-benzyloxycarbonyl-L-lysyl-glycyl-L-arginine 4-nitroanilide |
| factor IXa | Bos taurus | N-benzyloxycarbonyl-L-lysyl-L-phenylalanyl-L-arginine 4-nitroanilide | — | — | 0.0037 | pH 7.5, 25 °C | Open record: factor IXa, N-benzyloxycarbonyl-L-lysyl-L-phenylalanyl-L-arginine 4-nitroanilide |
| factor IXa | Bos taurus | N-benzyloxycarbonyl-L-prolyl-glycyl-L-arginine 4-nitroanilide | — | — | 7 × 10⁻⁵ | pH 7.5, 25 °C | Open record: factor IXa, N-benzyloxycarbonyl-L-prolyl-glycyl-L-arginine 4-nitroanilide |
| factor IXa | Bos taurus | N-benzyloxycarbonyl-L-seryl-glycyl-L-arginine 4-nitroanilide | — | — | 0.0017 | pH 7.5, 25 °C | Open record: factor IXa, N-benzyloxycarbonyl-L-seryl-glycyl-L-arginine 4-nitroanilide |
| factor IXa | Bos taurus | N-benzyloxycarbonyl-L-seryl-L-phenylalanyl-L-arginine 4-nitroanilide | — | — | 8.5 × 10⁻⁴ | pH 7.5, 25 °C | Open record: factor IXa, N-benzyloxycarbonyl-L-seryl-L-phenylalanyl-L-arginine 4-nitroanilide |
| factor Xa | Bos taurus | N-benzyloxycarbonyl-L-alanyl-glycyl-L-arginine 4-nitroanilide | 95 | 5.2 | 18 | pH 7.5, 25 °C | Open record: factor Xa, N-benzyloxycarbonyl-L-alanyl-glycyl-L-arginine 4-nitroanilide |
| factor Xa | Bos taurus | N-benzyloxycarbonyl-L-alanyl-L-phenylalanyl-L-arginine 4-nitroanilide | 1.8 | 0.24 | 7.5 | pH 7.5, 25 °C | Open record: factor Xa, N-benzyloxycarbonyl-L-alanyl-L-phenylalanyl-L-arginine 4-nitroanilide |
| factor Xa | Bos taurus | N-benzyloxycarbonyl-L-alpha-glutamyl-glycyl-L-arginine 4-nitroanilide | 433 | 11 | 39 | pH 7.5, 25 °C | Open record: factor Xa, N-benzyloxycarbonyl-L-alpha-glutamyl-glycyl-L-arginine 4-nitroanilide |
| factor Xa | Bos taurus | N-benzyloxycarbonyl-L-alpha-glutamyl-L-phenylalanyl-L-arginine 4-nitroanilide | 1 | 0.17 | 5.9 | pH 7.5, 25 °C | Open record: factor Xa, N-benzyloxycarbonyl-L-alpha-glutamyl-L-phenylalanyl-L-arginine 4-nitroanilide |
| factor Xa | Bos taurus | N-benzyloxycarbonyl-L-asparaginyl-glycyl-L-arginine 4-nitroanilide | 95 | 3.4 | 28 | pH 7.5, 25 °C | Open record: factor Xa, N-benzyloxycarbonyl-L-asparaginyl-glycyl-L-arginine 4-nitroanilide |
| factor Xa | Bos taurus | N-benzyloxycarbonyl-L-asparaginyl-L-phenylalanyl-L-arginine 4-nitroanilide | 20 | 2.1 | 9.5 | pH 7.5, 25 °C | Open record: factor Xa, N-benzyloxycarbonyl-L-asparaginyl-L-phenylalanyl-L-arginine 4-nitroanilide |
| factor Xa | Bos taurus | N-benzyloxycarbonyl-L-lysyl-glycyl-L-arginine 4-nitroanilide | 78 | 6.2 | 13 | pH 7.5, 25 °C | Open record: factor Xa, N-benzyloxycarbonyl-L-lysyl-glycyl-L-arginine 4-nitroanilide |
| factor Xa | Bos taurus | N-benzyloxycarbonyl-L-lysyl-L-phenylalanyl-L-arginine 4-nitroanilide | 0.58 | 0.24 | 2.4 | pH 7.5, 25 °C | Open record: factor Xa, N-benzyloxycarbonyl-L-lysyl-L-phenylalanyl-L-arginine 4-nitroanilide |
| factor Xa | Bos taurus | N-benzyloxycarbonyl-L-phenylalanyl-glycyl-L-arginine 4-nitroanilide | 152 | 4.5 | 34 | pH 7.5, 25 °C | Open record: factor Xa, N-benzyloxycarbonyl-L-phenylalanyl-glycyl-L-arginine 4-nitroanilide |
| factor Xa | Bos taurus | N-benzyloxycarbonyl-L-phenylalanyl-L-phenylalanyl-L-arginine 4-nitroanilide | 0.43 | 0.038 | 11 | pH 7.5, 25 °C | Open record: factor Xa, N-benzyloxycarbonyl-L-phenylalanyl-L-phenylalanyl-L-arginine 4-nitroanilide |
| factor Xa | Bos taurus | N-benzyloxycarbonyl-L-prolyl-glycyl-L-arginine 4-nitroanilide | 121 | 16 | 7.8 | pH 7.5, 25 °C | Open record: factor Xa, N-benzyloxycarbonyl-L-prolyl-glycyl-L-arginine 4-nitroanilide |
| factor Xa | Bos taurus | N-benzyloxycarbonyl-L-prolyl-L-phenylalanyl-L-arginine 4-nitroanilide | 1.1 | 0.99 | 1.1 | pH 7.5, 25 °C | Open record: factor Xa, N-benzyloxycarbonyl-L-prolyl-L-phenylalanyl-L-arginine 4-nitroanilide |
| factor Xa | Bos taurus | N-benzyloxycarbonyl-L-seryl-glycyl-L-arginine 4-nitroanilide | — | — | 29 | pH 7.5, 25 °C | Open record: factor Xa, N-benzyloxycarbonyl-L-seryl-glycyl-L-arginine 4-nitroanilide |
| factor Xa | Bos taurus | N-benzyloxycarbonyl-L-seryl-L-phenylalanyl-L-arginine 4-nitroanilide | 7.5 | 0.94 | 8 | pH 7.5, 25 °C | Open record: factor Xa, N-benzyloxycarbonyl-L-seryl-L-phenylalanyl-L-arginine 4-nitroanilide |
| factor XIa | Bos taurus | N-benzyloxycarbonyl-L-alanyl-glycyl-L-arginine 4-nitroanilide | — | — | 1.4 | pH 7.5, 25 °C | Open record: factor XIa, N-benzyloxycarbonyl-L-alanyl-glycyl-L-arginine 4-nitroanilide |
| factor XIa | Bos taurus | N-benzyloxycarbonyl-L-alanyl-L-phenylalanyl-L-arginine 4-nitroanilide | — | — | 1.6 | pH 7.5, 25 °C | Open record: factor XIa, N-benzyloxycarbonyl-L-alanyl-L-phenylalanyl-L-arginine 4-nitroanilide |
| factor XIa | Bos taurus | N-benzyloxycarbonyl-L-alpha-glutamyl-glycyl-L-arginine 4-nitroanilide | 12 | 2.9 | 4.1 | pH 7.5, 25 °C | Open record: factor XIa, N-benzyloxycarbonyl-L-alpha-glutamyl-glycyl-L-arginine 4-nitroanilide |
| factor XIa | Bos taurus | N-benzyloxycarbonyl-L-alpha-glutamyl-L-phenylalanyl-L-arginine 4-nitroanilide | 3.8 | 3.8 | 1 | pH 7.5, 25 °C | Open record: factor XIa, N-benzyloxycarbonyl-L-alpha-glutamyl-L-phenylalanyl-L-arginine 4-nitroanilide |
| factor XIa | Bos taurus | N-benzyloxycarbonyl-L-asparaginyl-glycyl-L-arginine 4-nitroanilide | 21 | 14 | 1.5 | pH 7.5, 25 °C | Open record: factor XIa, N-benzyloxycarbonyl-L-asparaginyl-glycyl-L-arginine 4-nitroanilide |
| factor XIa | Bos taurus | N-benzyloxycarbonyl-L-asparaginyl-L-phenylalanyl-L-arginine 4-nitroanilide | 2 | 0.71 | 2.8 | pH 7.5, 25 °C | Open record: factor XIa, N-benzyloxycarbonyl-L-asparaginyl-L-phenylalanyl-L-arginine 4-nitroanilide |
| factor XIa | Bos taurus | N-benzyloxycarbonyl-L-lysyl-glycyl-L-arginine 4-nitroanilide | 21 | 12 | 1.8 | pH 7.5, 25 °C | Open record: factor XIa, N-benzyloxycarbonyl-L-lysyl-glycyl-L-arginine 4-nitroanilide |
| factor XIa | Bos taurus | N-benzyloxycarbonyl-L-lysyl-L-phenylalanyl-L-arginine 4-nitroanilide | 2.5 | 2.7 | 0.93 | pH 7.5, 25 °C | Open record: factor XIa, N-benzyloxycarbonyl-L-lysyl-L-phenylalanyl-L-arginine 4-nitroanilide |
| factor XIa | Bos taurus | N-benzyloxycarbonyl-L-phenylalanyl-glycyl-L-arginine 4-nitroanilide | — | — | 3.8 | pH 7.5, 25 °C | Open record: factor XIa, N-benzyloxycarbonyl-L-phenylalanyl-glycyl-L-arginine 4-nitroanilide |
| factor XIa | Bos taurus | N-benzyloxycarbonyl-L-phenylalanyl-L-phenylalanyl-L-arginine 4-nitroanilide | 12 | 15 | 0.81 | pH 7.5, 25 °C | Open record: factor XIa, N-benzyloxycarbonyl-L-phenylalanyl-L-phenylalanyl-L-arginine 4-nitroanilide |
| factor XIa | Bos taurus | N-benzyloxycarbonyl-L-prolyl-glycyl-L-arginine 4-nitroanilide | 3.3 | 8.4 | 0.39 | pH 7.5, 25 °C | Open record: factor XIa, N-benzyloxycarbonyl-L-prolyl-glycyl-L-arginine 4-nitroanilide |
| factor XIa | Bos taurus | N-benzyloxycarbonyl-L-prolyl-L-phenylalanyl-L-arginine 4-nitroanilide | — | — | 0.29 | pH 7.5, 25 °C | Open record: factor XIa, N-benzyloxycarbonyl-L-prolyl-L-phenylalanyl-L-arginine 4-nitroanilide |
| factor XIa | Bos taurus | N-benzyloxycarbonyl-L-seryl-glycyl-L-arginine 4-nitroanilide | 7.1 | 2.4 | 3 | pH 7.5, 25 °C | Open record: factor XIa, N-benzyloxycarbonyl-L-seryl-glycyl-L-arginine 4-nitroanilide |
| factor XIa | Bos taurus | N-benzyloxycarbonyl-L-seryl-L-phenylalanyl-L-arginine 4-nitroanilide | 4.5 | 1.2 | 3.8 | pH 7.5, 25 °C | Open record: factor XIa, N-benzyloxycarbonyl-L-seryl-L-phenylalanyl-L-arginine 4-nitroanilide |
| thrombin | Bos taurus | N-benzyloxycarbonyl-L-alanyl-glycyl-L-arginine 4-nitroanilide | 0.92 | 0.24 | 3.8 | pH 7.5, 25 °C | Open record: thrombin, N-benzyloxycarbonyl-L-alanyl-glycyl-L-arginine 4-nitroanilide |
| thrombin | Bos taurus | N-benzyloxycarbonyl-L-alanyl-L-phenylalanyl-L-arginine 4-nitroanilide | 0.32 | 0.51 | 0.63 | pH 7.5, 25 °C | Open record: thrombin, N-benzyloxycarbonyl-L-alanyl-L-phenylalanyl-L-arginine 4-nitroanilide |
| thrombin | Bos taurus | N-benzyloxycarbonyl-L-alpha-glutamyl-glycyl-L-arginine 4-nitroanilide | 1.3 | 0.52 | 2.5 | pH 7.5, 25 °C | Open record: thrombin, N-benzyloxycarbonyl-L-alpha-glutamyl-glycyl-L-arginine 4-nitroanilide |
| thrombin | Bos taurus | N-benzyloxycarbonyl-L-alpha-glutamyl-L-phenylalanyl-L-arginine 4-nitroanilide | 0.18 | 0.33 | 1.8 | pH 7.5, 25 °C | Open record: thrombin, N-benzyloxycarbonyl-L-alpha-glutamyl-L-phenylalanyl-L-arginine 4-nitroanilide |
| thrombin | Bos taurus | N-benzyloxycarbonyl-L-asparaginyl-glycyl-L-arginine 4-nitroanilide | 0.41 | 0.22 | 1.9 | pH 7.5, 25 °C | Open record: thrombin, N-benzyloxycarbonyl-L-asparaginyl-glycyl-L-arginine 4-nitroanilide |
| thrombin | Bos taurus | N-benzyloxycarbonyl-L-asparaginyl-L-phenylalanyl-L-arginine 4-nitroanilide | 0.7 | 5.7 | 8 | pH 7.5, 25 °C | Open record: thrombin, N-benzyloxycarbonyl-L-asparaginyl-L-phenylalanyl-L-arginine 4-nitroanilide |
| thrombin | Bos taurus | N-benzyloxycarbonyl-L-lysyl-glycyl-L-arginine 4-nitroanilide | 2.3 | 0.22 | 10 | pH 7.5, 25 °C | Open record: thrombin, N-benzyloxycarbonyl-L-lysyl-glycyl-L-arginine 4-nitroanilide |
| thrombin | Bos taurus | N-benzyloxycarbonyl-L-lysyl-L-phenylalanyl-L-arginine 4-nitroanilide | 0.18 | 1.3 | 7.2 | pH 7.5, 25 °C | Open record: thrombin, N-benzyloxycarbonyl-L-lysyl-L-phenylalanyl-L-arginine 4-nitroanilide |
| thrombin | Bos taurus | N-benzyloxycarbonyl-L-phenylalanyl-glycyl-L-arginine 4-nitroanilide | 3.5 | 0.49 | 7.1 | pH 7.5, 25 °C | Open record: thrombin, N-benzyloxycarbonyl-L-phenylalanyl-glycyl-L-arginine 4-nitroanilide |
| thrombin | Bos taurus | N-benzyloxycarbonyl-L-phenylalanyl-L-phenylalanyl-L-arginine 4-nitroanilide | 0.15 | 0.026 | 5.8 | pH 7.5, 25 °C | Open record: thrombin, N-benzyloxycarbonyl-L-phenylalanyl-L-phenylalanyl-L-arginine 4-nitroanilide |
| thrombin | Bos taurus | N-benzyloxycarbonyl-L-prolyl-glycyl-L-arginine 4-nitroanilide | 0.91 | 0.16 | 5.7 | pH 7.5, 25 °C | Open record: thrombin, N-benzyloxycarbonyl-L-prolyl-glycyl-L-arginine 4-nitroanilide |
| thrombin | Bos taurus | N-benzyloxycarbonyl-L-seryl-glycyl-L-arginine 4-nitroanilide | 2.3 | 3.8 | 6.1 | pH 7.5, 25 °C | Open record: thrombin, N-benzyloxycarbonyl-L-seryl-glycyl-L-arginine 4-nitroanilide |
| thrombin | Bos taurus | N-benzyloxycarbonyl-L-seryl-L-phenylalanyl-L-arginine 4-nitroanilide | 1.2 | 0.18 | 6.7 | pH 7.5, 25 °C | Open record: thrombin, N-benzyloxycarbonyl-L-seryl-L-phenylalanyl-L-arginine 4-nitroanilide |
| β-factor XIIa | Homo sapiens | N-benzyloxycarbonyl-glycyl-L-arginine S-isobutyl thioester (SCH2CH(CH3)2) | 43 | 0.036 | 1.2 × 10³ | pH 7.5, 25 °C | Open record: β-factor XIIa, N-benzyloxycarbonyl-glycyl-L-arginine S-isobutyl thioester (SCH2CH(CH3)2) |
| β-factor XIIa | Homo sapiens | N-benzyloxycarbonyl-L-alanyl-glycyl-L-arginine 4-nitroanilide | 25 | 3.9 | 6.5 | pH 7.5, 25 °C | Open record: β-factor XIIa, N-benzyloxycarbonyl-L-alanyl-glycyl-L-arginine 4-nitroanilide |
| β-factor XIIa | Homo sapiens | N-benzyloxycarbonyl-L-alanyl-L-arginine S-benzyl thioester (SCH2C6H5) | 15 | 0.012 | 1.3 × 10³ | pH 7.5, 25 °C | Open record: β-factor XIIa, N-benzyloxycarbonyl-L-alanyl-L-arginine S-benzyl thioester (SCH2C6H5) |
| β-factor XIIa | Homo sapiens | N-benzyloxycarbonyl-L-alanyl-L-arginine S-isobutyl thioester (SCH2CH(CH3)2) | 14 | 0.034 | 410 | pH 7.5, 25 °C | Open record: β-factor XIIa, N-benzyloxycarbonyl-L-alanyl-L-arginine S-isobutyl thioester (SCH2CH(CH3)2) |
| β-factor XIIa | Homo sapiens | N-benzyloxycarbonyl-L-alanyl-L-phenylalanyl-L-arginine 4-nitroanilide | 34.6 | 1.5 | 23 | pH 7.5, 25 °C | Open record: β-factor XIIa, N-benzyloxycarbonyl-L-alanyl-L-phenylalanyl-L-arginine 4-nitroanilide |
| β-factor XIIa | Homo sapiens | N-benzyloxycarbonyl-L-alpha-glutamyl-glycyl-L-arginine 4-nitroanilide | — | — | 5.9 | pH 7.5, 25 °C | Open record: β-factor XIIa, N-benzyloxycarbonyl-L-alpha-glutamyl-glycyl-L-arginine 4-nitroanilide |
| β-factor XIIa | Homo sapiens | N-benzyloxycarbonyl-L-alpha-glutamyl-L-arginine S-isobutyl thioester (SCH2CH(CH3)2) | 9.2 | 0.15 | 61 | pH 7.5, 25 °C | Open record: β-factor XIIa, N-benzyloxycarbonyl-L-alpha-glutamyl-L-arginine S-isobutyl thioester (SCH2CH(CH3)2) |
| β-factor XIIa | Homo sapiens | N-benzyloxycarbonyl-L-alpha-glutamyl-L-phenylalanyl-L-arginine 4-nitroanilide | — | — | 12 | pH 7.5, 25 °C | Open record: β-factor XIIa, N-benzyloxycarbonyl-L-alpha-glutamyl-L-phenylalanyl-L-arginine 4-nitroanilide |
| β-factor XIIa | Homo sapiens | N-benzyloxycarbonyl-L-arginine S-isobutyl thioester (SCH2CH(CH3)2) | 22 | 0.103 | 210 | pH 7.5, 25 °C | Open record: β-factor XIIa, N-benzyloxycarbonyl-L-arginine S-isobutyl thioester (SCH2CH(CH3)2) |
| β-factor XIIa | Homo sapiens | N-benzyloxycarbonyl-L-asparaginyl-glycyl-L-arginine 4-nitroanilide | 18 | 2.7 | 6.6 | pH 7.5, 25 °C | Open record: β-factor XIIa, N-benzyloxycarbonyl-L-asparaginyl-glycyl-L-arginine 4-nitroanilide |
| β-factor XIIa | Homo sapiens | N-benzyloxycarbonyl-L-asparaginyl-L-phenylalanyl-L-arginine 4-nitroanilide | 23 | 0.66 | 35 | pH 7.5, 25 °C | Open record: β-factor XIIa, N-benzyloxycarbonyl-L-asparaginyl-L-phenylalanyl-L-arginine 4-nitroanilide |
| β-factor XIIa | Homo sapiens | N-benzyloxycarbonyl-L-lysyl-glycyl-L-arginine 4-nitroanilide | 23 | 0.7 | 32 | pH 7.5, 25 °C | Open record: β-factor XIIa, N-benzyloxycarbonyl-L-lysyl-glycyl-L-arginine 4-nitroanilide |
| β-factor XIIa | Homo sapiens | N-benzyloxycarbonyl-L-lysyl-L-arginine S-isobutyl thioester (SCH2CH(CH3)2) | 15 | 0.054 | 280 | pH 7.5, 25 °C | Open record: β-factor XIIa, N-benzyloxycarbonyl-L-lysyl-L-arginine S-isobutyl thioester (SCH2CH(CH3)2) |
| β-factor XIIa | Homo sapiens | N-benzyloxycarbonyl-L-lysyl-L-phenylalanyl-L-arginine 4-nitroanilide | 23 | 0.16 | 140 | pH 7.5, 25 °C | Open record: β-factor XIIa, N-benzyloxycarbonyl-L-lysyl-L-phenylalanyl-L-arginine 4-nitroanilide |
| β-factor XIIa | Homo sapiens | N-benzyloxycarbonyl-L-methionyl-L-arginine S-isobutyl thioester (SCH2CH(CH3)2) | 2.5 | 0.019 | 130 | pH 7.5, 25 °C | Open record: β-factor XIIa, N-benzyloxycarbonyl-L-methionyl-L-arginine S-isobutyl thioester (SCH2CH(CH3)2) |
| β-factor XIIa | Homo sapiens | N-benzyloxycarbonyl-L-phenylalanyl-glycyl-L-arginine 4-nitroanilide | 14 | 8.2 | 1.7 | pH 7.5, 25 °C | Open record: β-factor XIIa, N-benzyloxycarbonyl-L-phenylalanyl-glycyl-L-arginine 4-nitroanilide |
| β-factor XIIa | Homo sapiens | N-benzyloxycarbonyl-L-phenylalanyl-L-arginine S-isobutyl thioester (SCH2CH(CH3)2) | 8.3 | 0.006 | 1.4 × 10³ | pH 7.5, 25 °C | Open record: β-factor XIIa, N-benzyloxycarbonyl-L-phenylalanyl-L-arginine S-isobutyl thioester (SCH2CH(CH3)2) |
| β-factor XIIa | Homo sapiens | N-benzyloxycarbonyl-L-phenylalanyl-L-phenylalanyl-L-arginine 4-nitroanilide | — | — | 19 | pH 7.5, 25 °C | Open record: β-factor XIIa, N-benzyloxycarbonyl-L-phenylalanyl-L-phenylalanyl-L-arginine 4-nitroanilide |
| β-factor XIIa | Homo sapiens | N-benzyloxycarbonyl-L-prolyl-glycyl-L-arginine 4-nitroanilide | 9.2 | 6.7 | 1.4 | pH 7.5, 25 °C | Open record: β-factor XIIa, N-benzyloxycarbonyl-L-prolyl-glycyl-L-arginine 4-nitroanilide |
| β-factor XIIa | Homo sapiens | N-benzyloxycarbonyl-L-prolyl-L-arginine S-isobutyl thioester (SCH2CH(CH3)2) | 8.3 | 0.036 | 230 | pH 7.5, 25 °C | Open record: β-factor XIIa, N-benzyloxycarbonyl-L-prolyl-L-arginine S-isobutyl thioester (SCH2CH(CH3)2) |
| β-factor XIIa | Homo sapiens | N-benzyloxycarbonyl-L-prolyl-L-phenylalanyl-L-arginine 4-nitroanilide | — | — | 0.3 | pH 7.5, 25 °C | Open record: β-factor XIIa, N-benzyloxycarbonyl-L-prolyl-L-phenylalanyl-L-arginine 4-nitroanilide |
| β-factor XIIa | Homo sapiens | N-benzyloxycarbonyl-L-seryl-glycyl-L-arginine 4-nitroanilide | — | — | 5.1 | pH 7.5, 25 °C | Open record: β-factor XIIa, N-benzyloxycarbonyl-L-seryl-glycyl-L-arginine 4-nitroanilide |
| β-factor XIIa | Homo sapiens | N-benzyloxycarbonyl-L-seryl-L-arginine S-isobutyl thioester (SCH2CH(CH3)2) | 13 | 0.056 | 230 | pH 7.5, 25 °C | Open record: β-factor XIIa, N-benzyloxycarbonyl-L-seryl-L-arginine S-isobutyl thioester (SCH2CH(CH3)2) |
| β-factor XIIa | Homo sapiens | N-benzyloxycarbonyl-L-seryl-L-phenylalanyl-L-arginine 4-nitroanilide | 28 | 0.96 | 29 | pH 7.5, 25 °C | Open record: β-factor XIIa, N-benzyloxycarbonyl-L-seryl-L-phenylalanyl-L-arginine 4-nitroanilide |
| β-factor XIIa | Homo sapiens | N-benzyloxycarbonyl-L-threonyl-L-arginine S-isobutyl thioester (SCH2CH(CH3)2) | 11 | 0.054 | 210 | pH 7.5, 25 °C | Open record: β-factor XIIa, N-benzyloxycarbonyl-L-threonyl-L-arginine S-isobutyl thioester (SCH2CH(CH3)2) |
| β-factor XIIa | Homo sapiens | N-benzyloxycarbonyl-L-valyl-L-arginine S-isobutyl thioester (SCH2CH(CH3)2) | 17 | 0.046 | 370 | pH 7.5, 25 °C | Open record: β-factor XIIa, N-benzyloxycarbonyl-L-valyl-L-arginine S-isobutyl thioester (SCH2CH(CH3)2) |
| β-factor XIIa | Homo sapiens | N-tert-butyloxycarbonyl-L-arginine S-benzyl thioester (SCH2C6H5) | 29 | 0.18 | 160 | pH 7.5, 25 °C | Open record: β-factor XIIa, N-tert-butyloxycarbonyl-L-arginine S-benzyl thioester (SCH2C6H5) |
| β-factor XIIa | Homo sapiens | N-tert-butyloxycarbonyl-L-arginine S-isobutyl thioester (SCH2CH(CH3)2) | 9.2 | 0.095 | 610 | pH 7.5, 25 °C | Open record: β-factor XIIa, N-tert-butyloxycarbonyl-L-arginine S-isobutyl thioester (SCH2CH(CH3)2) |